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hGPR91 antagonist 3
CAS No. 1314796-31-0
hGPR91 antagonist 3( —— )
Catalog No. M35675 CAS No. 1314796-31-0
hGPR91 antagonist 3 is an orally active, potent, and selective hGPR91 antagonist. hGPR91 antagonist 3 is used to study hypertension, autoimmune diseases, and retinal angiogenesis.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 226 | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NamehGPR91 antagonist 3
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NoteResearch use only, not for human use.
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Brief DescriptionhGPR91 antagonist 3 is an orally active, potent, and selective hGPR91 antagonist. hGPR91 antagonist 3 is used to study hypertension, autoimmune diseases, and retinal angiogenesis.
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DescriptionhGPR91 antagonist 3 (Compound 5g) is a potent and orally active GPR91 antagonist with IC50 of 35 nM and 135 nM, for human GPR91 and rat GPR91, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetGPR
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RecptorGPR
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Research Area——
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Indication——
Chemical Information
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CAS Number1314796-31-0
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Formula Weight458.41
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Molecular FormulaC23H18F4N4O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (218.15 mM; Ultrasonic (<80°C)
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SMILESO=C(NCC=1ON=C(C1)C=2C=CC(F)=C(C2)C(F)(F)F)CCCC=3N=C4N=CC=CC4=CC3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Bhuniya D, et al. Discovery of a potent and selective small molecule hGPR91 antagonist. Bioorg Med Chem Lett. 2011;21(12):3596-3602. ?
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